Estrace vs Premarin: Kala duwanaanshaha, isku ekaanshaha, iyo yaa adiga kuu fiican
Daroogada Vs. SaaxiibDulmarka daroogada & kala duwanaanshaha ugu weyn | Xaaladaha la daweeyay | Wax ku oolnimada | Caymiska caymiska iyo isbarbardhiga qiimaha | Dhibaatooyinka ay keento | Isdhexgalka daroogada | Digniinta | Su'aalaha
Haddii aad isku aragto astaamo caadada ka joogsada, sida holaca kulul, dhidid habeenkii , dhibaatooyinka hurdada, iyo qallaylka xubinta taranka haweenka, bixiyahaaga daryeelka caafimaadka ayaa laga yaabaa inuu xusay daaweynta badalida hormoonka ama daaweynta estrogen. Calaamadaha menopause-ka waxay dhacaan marka jirku sameeyo estrogen yar, sidaa darteed daawooyinka beddelaya estrogen waxay gacan ka geysan karaan hagaajinta astaamahan, waxayna sidoo kale gacan ka geystaan kahortagga lafo-beelka.
Haweenka ilmo galeenka leh, daaweynta hoormoonka waxaa ku jira estrogen iyo progesterone labadaba. Haweenka ilmo-galeenka leh, estrogen kaligiis ayaa kordhiya halista kansarka endometrial.
Haweenka aan ilmo galeenka lahayn (ee soo maray makaanka kaadi mareenka) uma baahna inay qaataan progesterone leh estrogen. Haweenkan waxay isticmaali karaan alaabada estrogen-ka kaliya sida Estrace ama Premarin.
Estrace iyo Premarin waa laba daawo magac oo caan ah oo loogu talagalay daaweynta calaamadaha menopause. Labada daroogoba waxaa ansixiyay Maamulka Cuntada iyo Dawooyinka ee Mareykanka (FDA). Waxay ku jiraan fasal dawooyin ah oo loo yaqaan estrogens waxaana sidoo kale loo yaqaan daaweynta hoormoonka beddelaadda. Waxaa lagu heli karaa qaabab kala duwan, oo ay ku jiraan kareemooyin iyo kiniinno. In kasta oo Estrace iyo Premarin labaduba ay kujiraan estrogen, haddana si sax ah iskuma mid aha. Sii wad akhriska si aad waxbadan uga barato Estrace iyo Premarin.
Waa maxay farqiga u dhexeeya Estrace iyo Premarin?
Estrace waxaa lagu heli karaa nooc ahaan iyo qaab guud waxaana ku jira maaddada estradiol . Estrace waxaa loo heli karaa sida kareemka estrogen ee xubinta taranka haweenka, iyo sidoo kale kiniin afka laga qaato.
Premarin waxaa loo heli karaa oo kaliya daawo magac caan ah. Waxay ka kooban tahay estrogens isku dhafan, oo laga nadiifiyey kaadi mareska uurka leh (sidaa awgeed magaca loo yaqaan 'Premarin- PREgnan MARes urINe'). Premarin waxaa loo heli karaa sida kareemka estrogen ee xubinta taranka dumarka, kiniin afka ah, ama cirbad.
| Farqiga ugu weyn ee u dhexeeya Estrace iyo Premarin | ||
|---|---|---|
| Estrace | Premarin | |
| Fasalka daroogada | Daaweynta beddelka estrogens / hoormoonka | Daaweynta beddelka estrogens / hoormoonka |
| Summad / astaan guud | Nooc iyo astaan guud | Summad |
| Waa maxay magaca guud? | Estradiol | Estrogens isku dhafan |
| Waa noocee (yada) daroogadu soo gasho? | Kiriimka siilka, kaniiniga afka | Kiriimka siilka, kaniiniga afka, cirbadeynta |
| Waa maxay qiyaasta caadiga ah? | Kareem: 2 ilaa 4 garaam oo si caadi ah maalin walba 1-2 usbuuc, ka dibna si tartiib tartiib ah hoos ugu dhig qiyaasta dayactirka ee 1 garaam 1-3 jeer asbuucii Kiniiniyada: way kala duwan yihiin | Kariim: 0.5 garaam oo siil ah laba jeer usbuucii Kiniiniyada: way kala duwan yihiin |
| Muddo intee le'eg ayaa daaweynta caadiga ah? | Kaladuwan | Kaladuwan |
| Ayaa si caadi ah u isticmaala daawada? | Haweenka dhalmada kadib, mararka qaarkood ragga calaamadaha qaarkood (hoos eeg) | Haweenka dhalmada kadib, mararka qaarkood ragga calaamadaha qaarkood (hoos eeg) |
Xaaladaha ay daweeyeen Estrace iyo Premarin
Kreemka 'Estrace cream' iyo 'Premarin cream' waxay daaweeyaan astaamo dhexdhexaad ah ama daran oo ah soo-baxa xubinta taranka haweenka iyo xubinta taranka (khafiifinta, qallajinta, iyo bararka) caadada awgeed.
Foomka kaniiniga, Estrace iyo Premarin waxay ku daaweeyaan xaalado kale oo kala duwan oo ku taxan jaantuska hoose.
| Xaaladda | Estrace | Premarin |
| Calaamado dhexdhexaad ah oo daran oo soo noqnoqda xubinta taranka haweenka / dayska xubinta taranka haweenka | Haa (kareem) | Haa (kareem) |
| Daaweynta hypoestrogenism sababtoo ah hypogonadism, castration, ama ugxansidaha ugxan-yarida | Haa (kiniin) | Haa (kiniin) |
| Daaweynta kansarka naasaha (loogu talagalay kaliya daaweynta) haweenka iyo ragga qaarkood ee qaba cudurka metastatic | Haa (kiniin) | Haa (kiniin) |
| Daaweynta kansarka qanjirka 'prostate' ee qanjirka 'prostate' (qanjirada oo keliya) | Haa (kiniin) | Haa (kiniin) |
| Ka-hortagga cudurka 'postmenopausal osteoporosis' ee haweenka halista sare ku jira, marka daawooyinka aan estrogen ahayn aysan ku habboonayn | Haa (kiniin) | Haa (kiniin) |
| Daaweynta xubinta taranka dumarka iyo kilurosis | Off-calaamadda | Haa (kareem) |
| Daaweynta dyspareunia dhexdhexaad ah ama daran (galmo xanuun leh) dhalmo-dayska awgeed | Off-calaamadda | Haa (kareem) |
| Daaweynta calaamadaha vasomotor ee dhexdhexaadka ah ama daran ee dhalmo-dayska | Haa (kiniin) | Haa (kiniin) |
Estrace ama Premarin waxtar badan ma leedahay?
Daraasadaha ayaa muujinaya marka la isbarbar dhigayo alaabada estrogen, estradiol (maaddada Estrace) iyo estrogens conjugated (maaddada ku jirta Premarin) ayaa si isku mid ah waxtar ugu leh daaweynta calaamadaha menopause. Kareemada siilka wax ku ool ah oo si fiican loogu dulqaatay.
Bixiyahaaga daryeel caafimaad ayaa go'aamin kara daawada kugu habboon adiga, iyadoo la tixgelinayo astaamahaaga, xaaladahaaga caafimaad, iyo taariikhdaada caafimaad.
Daboolida iyo qiimaha isbarbar dhiga Estrace iyo Premarin
Qorshayaasha caymiska caymiska iyo Medicare ayaa sida caadiga ah daboolaya Estrace iyo Premarin.
Nooca dawada guud ee dawada 'Estrace' ayaa loogu talagalay tuubada kareemka waxayna ku kacaysaa $ 36 haddii aad jeebka ka bixiso, laakiin adeegsiga tigidhada 'SingleCare' ee bilaashka ah waxay hoos ugu dhigi kartaa qiimaha ugu yaraan $ 6.
Dawada caadiga ah ee daawada loogu talagalay tuubada Premarin waxay ku kacaysaa $ 250 jeebkiisa. Kaarka SingleCare wuxuu hoos ugu dhigi karaa qiimaha ugu hooseeya $ 198.
Maaddaama qorshayaashu kala duwan yihiin, la xiriir bixiyaha caymiska si aad u hesho faahfaahinta caymiska.
| Estrace | Premarin | |
| Caadi ahaan caymiska ayaa daboolaya? | Haa | Haa |
| Caadi ahaan waxaa daboola Medicare Qaybta D? | Haa | Haa |
| Tirada | 1 tuubo | 1 tuubo |
| Bixinta lacagta caadiga ah ee 'Medicare' | $ 1- $ 36 | $ 2- $ 451 |
| Qiimaha SingleCare | $ 6 + | $ 198 + |
Waxyeelooyinka guud ee Estrace iyo Premarin
Saameynaha ugu caansan ee Estrace iyo kareemka Premarin waxaa ka mid ah falcelinta goobta laga sameeyo sida cuncunka, dheecaanka, dhiig baxa makaanka, iyo barar. Intaa waxaa sii dheer, madax xanuun iyo miskaha xanuun ayaa dhici kara. Boqolkiiba waxyeellooyinka kuma jiraan macluumaadka qoritaanka ee Estrace.
Dhibaatooyinka soo raaca ee caadiga ah ee Estrace iyo Premarin ee qaabka kiniiniga ah ayaa ka nidaam badan. Qaar ka mid ah dhibaatooyinkaas soo raaca waxaa ka mid ah caloosha ama dhabar xanuun, daciifnimo, barar, madax xanuun, calool istaag, gaas, lallabbo, miisaanka oo kordha, niyad jab, wareer, wareer, naasaha oo u nugul / xanuun / isbedel, iyo dheecaanka hoosta haweenka, dhiig bax, ama infekshinka khamiirka.
Tani ma aha liistada buuxda ee waxyeellooyinka. Dhibaatooyinka kale ee xun ayaa dhici kara. La tasho daryeel caafimaad bixiyahaaga si aad ugala hadasho dhibaatooyinka soo raaca ee la filayo, iyo sida wax looga qabto.
| Kareemka Estrace | Kareemka Premarin | |||
| Waxyeellada | Ma khuseysaa? | Joogtaynta | Ma khuseysaa? | Joogtaynta |
| Madax xanuun | Haa | % lama sheegin | Haa | 3-5% * |
| Xanuun miskaha | Haa | % lama sheegin | Haa | 4% |
| Cuncun | Haa | % lama sheegin | Haa | 1-2% |
| Dheecaanka siilka | Maaha | - | Haa | 3-4% |
| Dhiigbaxa siilka | Haa | % lama sheegin | Haa | 1-2% |
| Caabuq siilka ah | Haa | % lama sheegin | Haa | 1-2% |
| Infekshinka xubinta taranka haweenka / caabuqa khamiirka | Haa | % lama sheegin | Haa | 3-4% |
* waxay kuxirantahay inta jeer ee qiyaasta daawada
Xigasho: DailyMed ( Kareemka Estrace ),, DailyMed ( Kareemka Premarin )
Isdhexgalka daroogada ee Estrace iyo Premarin
Estrace ama Premarin waxaa saameyn ku yeelan kara daawooyinka qaarkood oo ay dheefshiido enzme loo yaqaan cytochrome-p 450 3A4. Daawooyinka xakameynaya enzyme-ka ayaa hoos u dhigi kara howsha jirka ee Estrace ama Premarin, taasoo la micno ah Estrace ama Premarin ayaa laga yaabaa inay jirka ku sii jiraan muddo dheer, taasoo keenta waxyeelo badan. Sidoo kale, daawooyinka kiciya enzyme-ka waxay sababi karaan in jidhku dhaqso u shaqeeyo Estrace ama Premarin, taasoo ka dhigaysa mid aan waxtar badan lahayn. La tasho bixiyahaaga daryeelka caafimaadka wixii ku saabsan isdhexgalka daroogada ee suurtogalka ah.
| Daroogada | Fasalka daroogada | Estrace | Premarin |
| Clarithromycin Erythromycin Casiirka canabka Itraconazole Ketoconazole Ritonavir | CYP3A4 enzyme inhibitors | Suurtagal | Suurtagal |
| Carbamazepine Phenobarbital Rifampin Johannesört wort | CYP3A4 soo-saareyaasha enzyme | Suurtagal | Suurtagal |
Digniinta Estrace iyo Premarin
Estrace iyo Premarin waxay leeyihiin a digniinta sanduuqa , taas oo ah digniinta ugu xoogan ee ay u baahan tahay FDA. Sababtoo ah nuugista nidaamku waxay ku dhici kartaa kareemka Estrace ama kareemka Premarin, digniinta waxay khuseysaa dhammaan qaababka.
Estrogen keli ah:
- Isticmaalka estrogen keligiis (iyada oo aan lahayn progesin) haweeneyda ilmo-galeenka waxay kordhisaa halista kansarka endometrial. Ku darista progestin daaweynta estrogen waxay yareyn kartaa halista kansarka endometrial (laakiin waxay kordhin kartaa halista kansarka naasaha). Haweenka dhalmo-dayska ah ee dhiig-baxa aan caadiga ahayn waa in la tijaabiyaa si looga hortago xumaanta.
- Ha u isticmaalin estrogen kaligaa inaad ka hortagto wadne xanuunka ama waallida. Hindisaha Caafimaadka Haweenka (WHI) barasho waxay heleen halista sii kordheysa ee istaroogga iyo DVT (xinjirowga xididada dhiigga ee qotada dheer, ama xinjirowga dhiigga ee lugta) haweenka postmenopausal ee qaatay estrogen kaligood (progesin la'aan).
- Daraasadda ayaa sidoo kale muujisay halista sii kordheysa ee waallida ee haweenka postmenopausal ee qaatay estrogen kaligood.
Estrogen oo lagu daray progestin:
- Ha u isticmaalin estrogen oo lagu daro progestin si looga hortago cudurka wadnaha ama waallida. Daraasadda WHI waxay ogaatay khataro sare oo ah DVT, PE (sambabada sambabada), istaroog, iyo MI ee haweenka postmenopausal ee qaatay estrogen lagu daray progesin. Daraasadu waxay sidoo kale muujisay halista sare ee waallida ee haweenka postmenopausal ee qaatay estrogen iyo progesins.
- Daraasadda WHI waxay sidoo kale muujisay khatarta sii kordheysa ee kansarka naasaha ee ku dhaca estrogen oo lagu daray progestin.
Sidaa darteed, estrogens, iyada oo aan loo eegin haddii loo qoray ama aan lahayn progestins, waa in lagu qoro qiyaasta ugu hooseysa iyo muddada ugu gaaban. Kala hadal bixiyahaaga daryeelka caafimaadka halista iyo faa'iidooyinka noocyada kala duwan ee daaweynta beddelka hoormoonka.
Dhakhtarkaagu wuxuu ku siin doonaa talo caafimaad oo ku saabsan baaritaanka. Dhammaan haweenka waa inay maraan baaritaanka naasaha sanadlaha ah ee xirfadlaha daryeelka caafimaadka oo ay sameeyaan is-baaritaan bille ah. Dhammaan haweenka waa inay lahaadaan raajada naasaha oo ku saleysan da'da, arrimaha halista, iyo taariikhda.
Digniinaha kale ee Estrace iyo Premarin ayaa raaca.
Ha isticmaalin Estrace ama Premarin haddii aad leedahay:
- Dhiigbax aan caadi ahayn oo aan la aqoonsan
- Kansarka naasaha (loo yaqaan, looga shakisan yahay, ama taariikh)
- Neoplasia ku tiirsan estrogen (la yaqaan ama laga shakiyo)
- DVT ama sambabka wadnaha (firfircoon ama taariikh)
- Firfircoon ama taariikhda cudurka thromboembolic (istaroog, MI)
- Falcelin hore ee anaphylactic ee estrogen
- Cudurka beerka
- Cilladaha dhiig-baxa dhiigga
- Uurka (la yaqaan ama laga shakiyo)
Isku-darka daaweynta hoormoonka (estrogen plus progestin) ayaa kordhin kara halista kansarka ugxan-sidaha.
Haweenka dhalmada kadib ee qaata estrogen waxay leeyihiin kororka halista cudurka xameetida ee u baahan qalliinka.
Dadka qaata estrogens, dhibaatooyinka aragga ayaa ka dhacay. Raadso daaweyn degdeg ah haddii aad lumiso aragga (qayb ahaan ama dhammaystiran), aragga laba-laabma, indho-bararidda, ama dhanjafka.
Marar dhif ah, dareen-celinta xasaasiyadda ayaa dhacday. Haddii aad leedahay finan, cuncun, neefsashada oo dhib ku ah, matag, ama barar wejiga, bushimaha, carrabka, gacmaha, ama cagaha, raadi daryeel caafimaad oo degdeg ah isla markiiba. Daawada Estrogen waxaa laga yaabaa inay uga sii darto astaamaha cudurka anjioedema ee haweenka qaba cudurka anjioedema ee la iska dhaxlo.
Kala hadal bixiyahaaga daryeelka caafimaadka halistaas kahor intaadan qaadan daawada Estrace ama Premarin, si aad u ogaato in daawadu ay kuu nabad tahay iyo in kale.
Su'aalaha badanaa la isweydiiyo ee ku saabsan Estrace vs. Premarin
Waa maxay Estrace?
Estrace waa dawo lagu beddelo hoormoon ay ku jirto estradiol. Waxaa loo adeegsadaa tilmaamo kala duwan, badiyaa astaamaha menopause-ka. Estrace waxaa loo heli karaa inay tahay kareem afka laga qaato iyo sidoo kale kiniin afka laga qaato.
Waa maxay Premarin?
Premarin sidoo kale waa daawo lagu badalo hormoonka. Premarin waxaa ku jira estrogens isku dhafan. Waxaa loo adeegsadaa tilmaamo dhowr ah, badiyaa calaamadaha menopause. Premarin waxaa loo heli karaa sida kaniiniga afka, kareemka intravaginal, iyo cirbad.
Estrace iyo Premarin ma isku mid baa?
Estrace iyo Premarin waa isku mid, laakiin si sax ah iskuma mid aha. Macluumaadka kor ku xusan wuxuu qeexayaa farqiga u dhexeeya labada daawo.
Estrace ama Premarin ma ka fiican yihiin?
Labada daawoba waxay wax ku ool u yihiin daaweynta calaamadaha menopause, si kastaba ha noqotee, daawooyinkani waxay la yimaadaan waxyeelo iyo haliso. La hadal daryeel caafimaad bixiyahaaga si loo go'aamiyo haddii Estrace ama Premarin ay kugu habboon yihiin.
Ma isticmaali karaa Estrace ama Premarin inta aan uurka leeyahay?
Maya. Midkoodna daawo looma isticmaali karo uurka.
Ma ku isticmaali karaa Estrace ama Premarin aalkolo?
Cabitaanka aalkolo ee ay weheliso Estrace ama Premarin way awoodaa khatartaada kordhi kansarka naasaha. La tasho xirfadlahaaga daryeelka caafimaadka si aad uga hesho talo ku saabsan isticmaalka khamriga xaaladaha caafimaad ee aad qabto oo dhan.
Waa maxay bedelka ugu fiican ee Premarin?
Estrace waa bedel la mid ah Premarin. Daawooyinka kale ee ay kujiraan estrogen waxaa kamid ah Vivelle Dot Patch, Climara Patch, ama xubinta taranka dumarka si qaab ah oo ah kaniiniyada xubinta taranka ee Vagifem (kaniiniyada xubinta taranka haweenka oo lagu dabaqo codsadaha siilka) ama Estring Vaginal Ring. La hadal daryeel caafimaad bixiyahaaga si aad u aragto haddii mid ka mid ah daawooyinkaasi ay kugu habboon yihiin adiga.
Estrogen iyo estradiol ma isku waxbaa?
Estradiol waa nooc ka mid ah estrogen, hormoon haween ah. Dhammaan alaabada estradiol waa estrogen. Si kastaba ha noqotee, waxaa jira qaabab kale oo estrogen ah oo aan ahayn kaliya estradiol. Tusaale ahaan, estrogens conjugated (Premarin) waa nooc kale oo estrogen ah.
Premarin ma keenaa waallida?
Premarin (iyo Estrace) waxay leeyihiin digniin sanduuq ah oo ku saabsan waallida. Daraasadda Xusuusta WHI ee kor ku xusan waxay ogaatay halista sii kordheysa ee waallida ee haweenka postmenopausal ee qaatay estrogen kaligood ama estrogen oo leh progestin. Sidaa darteed, macluumaadka qoro waxay ku talinayaan in estrogen, ha ahaato kali ama ha la qaato progestin, waa in lagu qoro qiyaasta ugu yar iyo waqtiga ugu yar.
Estrace miyuu kordhiyaa heerarka estrogen?
Estrace (iyo Premarin) waxay kordhiyaan heerarka estrogen. Xitaa qaabka siilka, waxaa jira nuugid nidaamsan, iyo heerarka estrogen ayaa kordha. Bixiyahaaga daryeelka caafimaad ayaa go'aamin kara badeecada kuugu haboon adiga.











